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0.0092
(4-aminoquinazolin-2-yl)methyl 3-aminopyrazine-2-carboxylate
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0017
(4-oxo-3,4-dihydrothieno[3,2-d]pyrimidin-2-yl)methyl 2-(furan-2-yl)quinoline-4-carboxylate
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0049
1-(1H-pyrrol-2-yl)-2-[(thieno[2,3-d]pyrimidin-4-yl)oxy]ethan-1-one
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.013
1-(2-phenylpyrimidin-4-yl)-N-[(4-propoxyphenyl)methyl]piperidine-4-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0017
1-(3-chlorophenyl)-5-ethyl-N-(4H-1,2,4-triazol-3-yl)-1H-pyrazole-4-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.00011
1-[(2-chlorophenyl)methyl]-N-(4H-1,2,4-triazol-3-yl)-1H-pyrazole-4-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0058
1-[7-(3,4-dimethylbenzoyl)-2H-[1,3]dioxolo[4,5-g]quinolin-8-yl]piperidine-4-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0038
2-(1H-inden-2-yl)-5-[2-(1H-indol-3-yl)ethyl]-4-methyl-1H-pyrazolo[4,3-c]pyridine-3,6(2H,5H)-dione
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0011
2-(5-chlorothiophen-2-yl)-2-oxoethyl (3,4-dimethoxyphenyl)acetate
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0066
2-(8-fluoro-3,4-dihydroquinolin-1(2H)-yl)-N-(quinolin-5-yl)acetamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0045
2-oxo-2-(2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)ethyl 2-methylquinoline-4-carboxylate
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0053
2-oxo-2-(2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)ethyl 3-(cyclopropylsulfamoyl)thiophene-2-carboxylate
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0015 - 0.0034
2-oxo-2-(3-sulfamoylanilino)ethyl 2-(furan-2-yl)quinoline-4-carboxylate
0.0034
2-oxo-2-[(quinolin-5-yl)amino]ethyl 1-(5-carbamoylpyridin-2-yl)piperidine-4-carboxylate
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.00093
2-phenyl-7-(quinoline-6-carbonyl)-5,6,7,8-tetrahydropyrazolo[1,5-a]pyrido[4,3-d]pyrimidin-9(1H)-one
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0007
2-[(3,5-dichloropyridin-2-yl)amino]-2-oxoethyl 5,6-dihydro-4H-cyclopenta[b]thiophene-2-carboxylate
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0029
2-[(4-acetylbenzene-1-sulfonyl)amino]thiophene-3-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.00053
2-[(5-chloropyridin-2-yl)amino]-2-oxoethyl 2-(furan-2-yl)quinoline-4-carboxylate
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0014
2-[2-(1-methyl-2-phenyl-2,3-dihydro-1H-indol-3-yl)-2-oxoethyl]-1,3-dioxo-1,2,3,5,6,7-hexahydropyrrolo[1,2-c]pyrimidine-4-carbonitrile
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0019
2-[2-(3-chlorophenoxy)acetamido]thiophene-3-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0025
2-[2-(4-oxocinnolin-1(4H)-yl)acetamido]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0027
2-[3-(benzenesulfonyl)-7-methyl-4-oxo-1,8-naphthyridin-1(4H)-yl]-N-methyl-N-phenylacetamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.002
2-[5-[2-(methylamino)-1,3-thiazol-4-yl]thiophen-2-yl]acetamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.00031
3-(1H-pyrrol-1-yl)-N-[4-[(1,3-thiazol-2-yl)sulfamoyl]phenyl]benzamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0017
3-(4-methoxyphenyl)-7-[(1H-pyrrol-2-yl)methyl]-5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyrazine
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0087
3-oxo-N-(5,6,7,8-tetrahydronaphthalen-1-yl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0091
3-oxo-N-[1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl]-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0097
3-oxo-N-[[2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl]-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0018
4-((4-azidobenzyl)oxy)-N-(4-((octylamino)methyl)benzyl)thieno-[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.000085
4-oxo-N-(4-((pentylamino)methyl)benzyl)-3,4-dihydrothieno-[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.0011
4-oxo-N-(4-(piperidin-1-ylmethyl)benzyl)-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.0019
4-[(tetrazolo[1,5-b]pyridazin-6-yl)amino]benzamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0056
4-[3-(8-hydroxyimidazo[1,2-a]pyridin-2-yl)-2,5-dimethyl-1H-pyrrol-1-yl]benzene-1-sulfonamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0029
4-[3-(pyridin-4-yl)-1H-pyrazol-5-yl]thiomorpholine
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0025
5,7-dimethyl-N-(4H-1,2,4-triazol-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.00049
5-(5-methylthiophen-2-yl)thieno[2,3-d]pyrimidin-4(3H)-one
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0036
5-[2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-2-oxoethyl]-2-(3-fluorophenyl)-7-methyl-3-(1H-pyrrol-1-yl)-2,3,3a,5-tetrahydro-4H-pyrazolo[3,4-d]pyridazin-4-one
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.011
6-(2-[[(furan-2-yl)methyl]amino]-1,3-thiazol-4-yl)-3,4-dihydroquinolin-2(1H)-one
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0054
6-[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl][1,2,4]triazolo[4,3-a]pyridine
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.006
ethyl 4-[(3-cyano-6,7-dimethoxyquinolin-4-yl)amino]benzoate
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0028
N-(2-methoxy-5-methylphenyl)-N'-[1,2,4]triazolo[4,3-a]pyridin-3-ylurea
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.005
N-(3,4-dimethylphenyl)-5,6-dihydro-4H-cyclopenta[d][1,2]oxazole-3-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0047
N-(3-acetylphenyl)-N2-[5-chloro-2-(pyrrolidin-1-yl)phenyl]glycinamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0016
N-(3-carbamoyl-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)-4-chloropyridine-2-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.006
N-(3-carbamoylthiophen-2-yl)-2-(pyridin-4-yl)quinoline-4-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0021
N-(3-cyanothiophen-2-yl)-2-(furan-2-yl)quinoline-4-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.00072
N-(4-((((3s,5s,7s)-adamantan-1-yl)amino)methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.00045
N-(4-(((2-(2-(2-aminoethoxy)ethoxy)ethyl)amino)methyl)-benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.00021
N-(4-(((2-(2-ethoxyethoxy)ethyl)amino)methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.00011
N-(4-(((2-(2-hydroxyethoxy)ethyl)amino)methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.00008
N-(4-(((4-aminobutyl)amino)methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide dihydrochloride
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.0013
N-(4-(((5-(1,5-dihydroxy-4-oxo-1,4-dihydropyridine-2-carboxamido)pentyl)amino) methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.00011
N-(4-(((5-aminopentyl)amino)methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.00014
N-(4-(((7-aminohexyl)amino)methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.0007
N-(4-((1,5-dihydroxy-4-oxo-1,4-dihydropyridine-2-carboxamido)methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]-pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.0022
N-(4-((benzyl(ethyl)amino)methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.0022
N-(4-((benzyl(hexyl)amino)methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.012
N-(4-((benzyl(octyl)amino)methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.00013
N-(4-((benzylamino)methyl)benzyl)-4-oxo-3,4-dihydrothieno-[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.00015
N-(4-((butylamino)methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.00049
N-(4-((cyclohexyl(ethyl)amino)methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.00079
N-(4-((cyclohexylamino)methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.000025
N-(4-((decylamino)methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.00073
N-(4-((diethylamino)methyl)benzyl)-4-oxo-3,4-dihydrothieno-[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.00038
N-(4-((dodecylamino)methyl)benzyl)-4-oxo-3,4-dihydrothieno-[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.00037
N-(4-((ethyl(octyl)amino)methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.000024
N-(4-((octylamino)methyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.003
N-(4-(morpholinomethyl)benzyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
0.0013
N-([1-[3-(pyridin-4-yl)-1H-pyrazol-5-yl]piperidin-4-yl]methyl)-1H-indole-2-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.01
N-([2-[(morpholin-4-yl)methyl]phenyl]methyl)-2-(thiophene-2-carbonyl)benzamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.00018
N-([4-[(4-aminopiperidin-1-yl)methyl]phenyl]methyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-5-carboxamide
Pseudomonas aeruginosa
-
pH 8.0, 37°C
-
0.0043
N-methyl-1-[2-([[2-(pyridin-3-yl)quinazolin-4-yl]amino]methyl)phenyl]methanesulfonamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0062
N-methyl-N-[(oxan-4-yl)methyl]-2-(thiophen-3-yl)acetamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0013
N-methyl-N-[[2-(pyrrolidin-1-yl)phenyl]methyl]-3-(1H-pyrrol-1-yl)benzamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0039
N-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]quinoline-6-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0029
N-[1-[3-(pyridin-4-yl)-1H-pyrazol-5-yl]piperidin-3-yl]-1H-indole-2-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.012
N-[1-[3-(pyridin-4-yl)-1H-pyrazol-5-yl]piperidin-3-yl]-2-(thiophen-2-yl)acetamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0068
N-[2-oxo-2-[(1,3,5-trimethyl-4,5-dihydro-1H-pyrazol-4-yl)amino]ethyl]-5,6-dihydro-4H-cyclopenta[b]thiophene-2-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0087
N-[3-(pyridin-4-yl)-1,2-oxazol-5-yl]-5,6,7,8-tetrahydronaphthalene-2-sulfonamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0021
N-[3-([1,3]thiazolo[5,4-b]pyridin-2-yl)phenyl]quinoline-2-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.014
N-[3-[(3-fluoro-4-methylphenyl)carbamoyl]phenyl]-1-([1,3]thiazolo[5,4-b]pyridin-2-yl)piperidine-3-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0019
N-[4-(2-amino-2-oxoethyl)-1,3-thiazol-2-yl]-3-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)propanamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0031
N-[4-chloro-3-(pyrrolidine-1-sulfonyl)phenyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.001
N-[[4-(piperidine-1-carbonyl)phenyl]methyl]-2-(thiophene-2-carbonyl)benzamide
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0083
sinefungin
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0091
suramin
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0059
[4-(hydroxymethyl)-2,8-diazaspiro[4.5]decan-2-yl][1-(4-methoxyphenyl)cyclohexyl]methanone
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0053
[5-(furan-2-yl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-2-yl]methyl pyrazine-2-carboxylate
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0015
2-oxo-2-(3-sulfamoylanilino)ethyl 2-(furan-2-yl)quinoline-4-carboxylate
Pseudomonas aeruginosa
pH and temperature not specified in the publication
0.0034
2-oxo-2-(3-sulfamoylanilino)ethyl 2-(furan-2-yl)quinoline-4-carboxylate
Pseudomonas aeruginosa
pH and temperature not specified in the publication