EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.17.3.2 | -999 |
- |
more |
inhibition kinetic analysis |
745094 |
1.17.3.2 | -999 |
- |
more |
inhibition kinetics |
685028, 685516, 685804, 745461 |
1.17.3.2 | 0.0000006 |
- |
2-[3-cyano-4-(2-methylpropoxy)phenyl]-4-methylthiazole-5-carboxylic acid |
25°C, pH 7.4, oxidized form of enzyme |
675736 |
1.17.3.2 | 0.0000031 |
- |
2-[3-cyano-4-(2-methylpropoxy)phenyl]-4-methylthiazole-5-carboxylic acid |
25°C, pH 7.4, reduced form of enzyme |
675736 |
1.17.3.2 | 0.0000475 |
- |
6-(N-benzoylamino)purine |
25°C, pH 7.5 |
675102 |
1.17.3.2 | 0.000094 |
- |
6-formylpterin |
- |
658067 |
1.17.3.2 | 0.00011 |
- |
2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-6-methoxy-4H-chromen-4-one |
pH 7.5, 25°C |
676739 |
1.17.3.2 | 0.00011 |
- |
5,7-dihydroxy-2-(4-methoxyphenyl)-4H-chromen-4-one |
pH 7.5, 25°C |
676739 |
1.17.3.2 | 0.00012 |
- |
5,7-dihydroxy-2-(3-hydroxy-4-methoxyphenyl)-4H-chromen-4-one |
pH 7.5, 25°C |
676739 |
1.17.3.2 | 0.00015 |
- |
2-(3,4-dihydroxy-5-methoxyphenyl)-5,7-dihydroxy-4H-chromen-4-one |
pH 7.5, 25°C |
676739 |