EC Number   |
Inhibitors |
Structure |
|---|
    2.1.1.5 | (2S,11RS)-5-thia-2,11-diamino-8,8-dimethyldodecanedioic acid |
more than 90% inhibition at 0.02 mM |
   |
| 2.1.1.5 | (2S,11RS)-5-thia-2,11-diaminododecanedioic acid |
about 60% inhibition at 0.02 mM |
|
| 2.1.1.5 | (2S,11S)-5,8-dithia-2,11-diaminododecanedioic acid |
about 60% inhibition at 0.02 mM |
|
| 2.1.1.5 | (2S,5RS,8RS,11S)-5,8-dithia-2,11-diaminododecanedioic acid 5,8-dioxide |
about 20% inhibition at 0.02 mM |
|
| 2.1.1.5 | (2S,8RS,11RS)-5-thia-2,11-diamino-8-methyldodecanedioic acid |
competitive, more than 90% inhibition at 0.02 mM |
|
| 2.1.1.5 | (R,S)-2-(3-amino-3-carboxy-propylsulfanyl)-benzoic acid |
ca. 43% inhibition at 0.02 mM |
|
| 2.1.1.5 | (R,S)-2-amino-4-(2-carboxy-ethyldisulfanyl)-butyric acid |
ca. 30% inhibition at 0.02 mM |
|
| 2.1.1.5 | (R,S)-2-amino-4-(2-carboxymethylsulfanyl-ethylsulfanyl)-butyric acid |
100% inhibition at 0.02 mM, very potent inhibitor and one of the strongest ever reported |
|
| 2.1.1.5 | (R,S)-2-amino-4-(2-carboxymethylsulfinyl-ethylsulfanyl)-butyric acid |
ca. 90% inhibition at 0.02 mM |
|
| 2.1.1.5 | (R,S)-2-amino-4-(2-phosphonomethoxy-ethylsulfanyl)-butyrate |
ca. 26% inhibition at 0.02 mM |
|
