Inhibitors | Comment | Organism | Structure |
---|---|---|---|
edrophonium | 33.7% inhibition at 0.1 mM, competitive inhibition | Electrophorus electricus | |
eserine | 20.1% inhibition at 0.1 mM | Electrophorus electricus | |
additional information | descending order of inhibitory potency is tacrine, edrophonium, neostigmine, eserine, pyridostigmine | Electrophorus electricus | |
neostigmine | 31.1% inhibition at 0.1 mM | Electrophorus electricus | |
pyridostigmine | 6.1% inhibition at 0.1 mM | Electrophorus electricus | |
tacrine | i.e. 9-amino-1,2,3,4-tetrahydroacridine hydrochloride, 54.2% inhibition at 0.1 mM, mixed-type inhibition | Electrophorus electricus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
acetylcholine + H2O | Electrophorus electricus | - |
acetate + choline | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Electrophorus electricus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
commercial preparation | - |
Electrophorus electricus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
acetylcholine + H2O | - |
Electrophorus electricus | acetate + choline | - |
? | |
additional information | activity detection using a capillary electrophoresis, EMMA, method, screening method development and optimization of experimental conditions, overview | Electrophorus electricus | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
AChE | - |
Electrophorus electricus |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
8 | - |
assay at | Electrophorus electricus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
additional information | - |
additional information | inhibition mechanism analysis and kinetics, overview | Electrophorus electricus |