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Literature summary for 3.1.1.7 extracted from

  • Musilova, L.; Kuca, K.; Jung, Y.S.; Jun, D.
    In vitro oxime-assisted reactivation of paraoxon-inhibited human acetylcholinesterase and butyrylcholinesterase (2009), Clin. Toxicol. (Phila.), 47, 545-550.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
paraoxon i.e. O,O-diethyl-O-4-nitrophenyl phosphate, the paraoxon-inhibited enzyme is reactivated by several compounds, kinetics, overview. Best reactivating compounds are obidoxime, K027, and trimedoxie Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
erythrocyte
-
Homo sapiens
-

Synonyms

Synonyms Comment Organism
AChE
-
Homo sapiens

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
25
-
assay at Homo sapiens

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
7.4
-
assay at Homo sapiens