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Literature summary for 3.1.1.7 extracted from

  • Agrawal, R.; Tyagi, E.; Shukla, R.; Nath, C.
    Effect of insulin and melatonin on acetylcholinesterase activity in the brain of amnesic mice (2008), Behav. Brain Res., 189, 381-386.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
donepezil AChE activity in detergent soluble fraction of scopolamine amnesic mice is inhibited by donepezil, insulin and melatonin with varying extent in different brain regions, whereas AChE activity in salt soluble fraction is not much affected, overview Mus musculus
Insulin AChE activity in detergent soluble fraction of scopolamine amnesic mice is inhibited by donepezil, insulin and melatonin with varying extent in different brain regions, whereas AChE activity in salt soluble fraction is not much affected, overview Mus musculus
Melatonin AChE activity in detergent soluble fraction of scopolamine amnesic mice is inhibited by donepezil, insulin and melatonin with varying extent in different brain regions, whereas AChE activity in salt soluble fraction is not much affected, overview Mus musculus

Organism

Organism UniProt Comment Textmining
Mus musculus
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Swiss adult male mice
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Source Tissue

Source Tissue Comment Organism Textmining
brain forebrain cholinergic neurons Mus musculus
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neuron forebrain cholinergic neurons Mus musculus
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Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
S-acetylthiocholine iodide + H2O detection with 5,5'-dithio-bis-2-nitrobenzoic acid, i.e. DTNB Mus musculus acetate + thiocholine iodide
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?

Synonyms

Synonyms Comment Organism
AChE
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Mus musculus

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
7
-
assay at Mus musculus