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Literature summary for 3.1.1.7 extracted from

  • Freitas, R.M.; Sousa, F.C.; Viana, G.S.; Fonteles, M.M.
    Acetylcholinesterase activities in hippocampus, frontal cortex and striatum of Wistar rats after pilocarpine-induced status epilepticus (2006), Neurosci. Lett., 399, 76-78.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
pilocarpine pilocarpine induction of status epilepticus leads to enzyme inhibition during seizures in the rat brain, overview Rattus norvegicus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
acetylcholine + H2O Rattus norvegicus
-
choline + acetate
-
?

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
Wistar rats
-

Source Tissue

Source Tissue Comment Organism Textmining
brain
-
Rattus norvegicus
-
frontal cortex
-
Rattus norvegicus
-
hippocampus
-
Rattus norvegicus
-
striatum
-
Rattus norvegicus
-

Specific Activity [micromol/min/mg]

Specific Activity Minimum [µmol/min/mg] Specific Activity Maximum [µmol/min/mg] Comment Organism
additional information
-
tissue-dependent activity with and without pilocarpine treatment, overview Rattus norvegicus

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
acetylcholine + H2O
-
Rattus norvegicus choline + acetate
-
?
acetylthiocholine + H2O
-
Rattus norvegicus thiocholine + acetate
-
?

Synonyms

Synonyms Comment Organism
AChE
-
Rattus norvegicus

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
37
-
assay at Rattus norvegicus

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
7
-
assay at Rattus norvegicus