Inhibitors | Comment | Organism | Structure |
---|---|---|---|
1-(3-bromo-4-methoxybenzene-1-sulfonyl)-3-[(1H-imidazol-1-yl)methyl]piperidine | - |
Homo sapiens | |
1-[3-(2-chloro-6-nitrophenyl)benzene-1-sulfonyl]-3-[(1H-imidazol-1-yl)methyl]piperidine | - |
Homo sapiens | |
4-[3-[(1H-imidazol-1-yl)methyl]piperidine-1-sulfonyl]-2,1,3-benzothiadiazole | - |
Homo sapiens | |
SYN 20028567 | nonsteroidal lead compound for aromatase inhibition | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
7-methoxy-4-trifluoromethyl coumarin + H2O + oxidized flavoprotein | - |
Homo sapiens | ? + O2 + reduced flavoprotein | - |
? |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.000006 | - |
pH not specified in the publication, temperature not specified in the publication | Homo sapiens | 1-(3-bromo-4-methoxybenzene-1-sulfonyl)-3-[(1H-imidazol-1-yl)methyl]piperidine | |
0.000007 | - |
pH not specified in the publication, temperature not specified in the publication | Homo sapiens | 4-[3-[(1H-imidazol-1-yl)methyl]piperidine-1-sulfonyl]-2,1,3-benzothiadiazole | |
0.000009 | - |
pH not specified in the publication, temperature not specified in the publication | Homo sapiens | 1-[3-(2-chloro-6-nitrophenyl)benzene-1-sulfonyl]-3-[(1H-imidazol-1-yl)methyl]piperidine | |
0.000009 | - |
pH not specified in the publication, temperature not specified in the publication | Homo sapiens | SYN 20028567 |