Activating Compound | Comment | Organism | Structure |
---|---|---|---|
MS-275 | - |
Renilla reniformis |
Cloned (Comment) | Organism |
---|---|
expression in HEK-293 cells or Grip-Tite 293 MSR cells | Renilla reniformis |
Protein Variants | Comment | Organism |
---|---|---|
T329G | no significant influence on enzyme activity | Renilla reniformis |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
N-benzyl-4-methylbenzenesulfonamide | inhibition of purified enzyme, inducing activity in cell-based assay | Renilla reniformis |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Renilla reniformis | - |
- |
- |
Purification (Comment) | Organism |
---|---|
- |
Renilla reniformis |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
coelenterazine-H + O2 | 5 microM, assay at pH 7.5 | Renilla reniformis | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
Renilla reniformis luciferase | - |
Renilla reniformis |
RLuc | - |
Renilla reniformis |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.5 | - |
assay at | Renilla reniformis |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0012 | - |
N-benzyl-4-methylbenzenesulfonamide | - |
Renilla reniformis |